Peptide
Peptides are short chains of between two and fifty amino acids, linked by peptide bonds. Chains of less than ten or fifteen amino acids are called oligopeptides, and include dipeptides, tripeptides, and tetrapeptides.
A polypeptide is a longer, continuous, unbranched peptide chain of up to approximately fifty amino acids. Hence, peptides fall under the broad chemical classes of biological polymers and oligomers, alongside nucleic acids, oligosaccharides, polysaccharides, and others.
A polypeptide that contains more than approximately fifty amino acids is known as a protein. Proteins consist of one or more polypeptides arranged in a biologically functional way, often bound to ligands such as coenzymes and cofactors, or to another protein or other macromolecule such as DNA or RNA, or to complex macromolecular assemblies.
Amino acids that have been incorporated into peptides are termed residues. A water molecule is released during formation of each amide bond. All peptides except cyclic peptides have an N-terminal and C-terminal residue at the end of the peptide.
Classes
Many kinds of peptides are known. They have been classified or categorized according to their sources and functions. According to the Handbook of Biologically Active Peptides, some groups of peptides include plant peptides, bacterial/antibiotic peptides, fungal peptides, invertebrate peptides, amphibian/skin peptides, venom peptides, cancer/anticancer peptides, vaccine peptides, immune/inflammatory peptides, brain peptides, endocrine peptides, ingestive peptides, gastrointestinal peptides, cardiovascular peptides, renal peptides, respiratory peptides, opiate peptides, neurotrophic peptides, and blood–brain peptides.Some ribosomal peptides are subject to proteolysis. These function, typically in higher organisms, as hormones and signaling molecules. Some organisms produce peptides as antibiotics, such as microcins and bacteriocins.
Peptides frequently have post-translational modifications such as phosphorylation, hydroxylation, sulfonation, palmitoylation, glycosylation, and disulfide formation. In general, peptides are linear, although lariat structures have been observed. More exotic manipulations do occur, such as racemization of L-amino acids to D-amino acids in platypus venom.
Nonribosomal peptides are assembled by enzymes, not the ribosome. A common non-ribosomal peptide is glutathione, a component of the antioxidant defenses of most aerobic organisms. Other nonribosomal peptides are most common in unicellular organisms, plants, and fungi and are synthesized by modular enzyme complexes called nonribosomal peptide synthetases.
These complexes are often laid out in a similar fashion, and they can contain many different modules to perform a diverse set of chemical manipulations on the developing product. These peptides are often cyclic and can have highly complex cyclic structures, although linear nonribosomal peptides are also common. Since the system is closely related to the machinery for building fatty acids and polyketides, hybrid compounds are often found. The presence of oxazoles or thiazoles often indicates that the compound was synthesized in this fashion.
are derived from animal milk or meat digested by proteolysis. In addition to containing small peptides, the resulting material includes fats, metals, salts, vitamins, and many other biological compounds. Peptones are used in nutrient media for growing bacteria and fungi.
Peptide fragments refer to fragments of proteins that are used to identify or quantify the source protein. Often these are the products of enzymatic degradation performed in the laboratory on a controlled sample, but can also be forensic or paleontological samples that have been degraded by natural effects.
Chemical synthesis
Example families
The peptide families in this section are ribosomal peptides, usually with hormonal activity. All of these peptides are synthesized by cells as longer "propeptides" or "proproteins" and truncated prior to exiting the cell. They are released into the bloodstream where they perform their signaling functions.Antimicrobial peptides
- Magainin family
- Cecropin family
- Cathelicidin family
- Defensin family
Tachykinin peptides
- Substance P
- Kassinin
- Neurokinin A
- Eledoisin
- Neurokinin B
Vasoactive intestinal peptides
- VIP
- PACAP Pituitary Adenylate Cyclase Activating Peptide
- Peptide PHI 27
- GHRH 1-24
- Glucagon
- Secretin
Pancreatic polypeptide-related peptides
- NPY
- PYY '
- APP '
- PPY Pancreatic PolYpeptide''
Opioid peptides
- Proopiomelanocortin peptides
- Enkephalin pentapeptides
- Prodynorphin peptides
Calcitonin peptides
- Calcitonin
- Amylin
- AGG01
Self-Assembling peptides
- Amphiphilic peptides
- Aromatic short peptides
- Biomimetic peptides
- Peptide dendrimers
Other peptides
- B-type Natriuretic Peptide - produced in the myocardium and useful in medical diagnosis
- Lactotripeptides - Lactotripeptides might reduce blood pressure, although the evidence is mixed.
- Peptidic components from traditional Chinese medicine Colla Corii Asini in hematopoiesis.
Terminology
Length
Several terms related to peptides have no strict length definitions, and there is often overlap in their usage.- A polypeptide is a single linear chain of many amino acids, held together by amide bonds.
- A protein consists of one or more polypeptides.
- An oligopeptide consists of only a few amino acids.
Number of amino acids
Peptides of defined length are named using IUPAC numerical multiplier prefixes.- A has one amino acid.
- A dipeptide has two amino acids.
- A tripeptide has three amino acids.
- A tetrapeptide has four amino acids.
- A pentapeptide has five amino acids.
- A hexapeptide has six amino acids.
- A heptapeptide has seven amino acids.
- An octapeptide has eight amino acids.
- A nonapeptide has nine amino acids.
- A decapeptide has ten amino acids.
Function
- A neuropeptide is a peptide that is active in association with neural tissue.
- A lipopeptide is a peptide that has a lipid connected to it, and pepducins are lipopeptides that interact with GPCRs.
- A peptide hormone is a peptide that acts as a hormone.
- A proteose is a mixture of peptides produced by the hydrolysis of proteins. The term is somewhat archaic.
- A peptidergic agent is a chemical which functions to directly modulate the peptide systems in the body or brain. An example is opioidergics, which are neuropeptidergics.