List of estrogen esters


This is a list of estrogen esters, or ester prodrugs of estrogens. It includes esters, as well as ethers, of steroidal estrogens like estradiol, estrone, and estriol and of nonsteroidal estrogens like the stilbestrols diethylstilbestrol and hexestrol.

Esters of steroidal estrogens

Estradiol esters

Marketed

Many esters of estradiol have been marketed, including the following major esters:
And the following less commonly used esters:
The following nitrogen mustard ester of estradiol is an cytostatic antineoplastic agent and has been marketed:
A few other estradiol esters which are notable but have not been marketed include:
The following cytostatic antineoplastic nitrogen mustard esters of estradiol have not been marketed:

Marketed

Esters of estrone that have been marketed include:
Other estrone esters which are notable but have not been marketed include:

Marketed

Esters of estriol that have been marketed include:
The following ester of estriol was never marketed:

Marketed

The following esters of ethinylestradiol exist and have been marketed:

Marketed

The following esters of other estrogens exist and have been marketed:

Marketed

A number of estrogen ethers also exist and have been marketed, including:
A few other estrogen ethers which are notable but have not been marketed include:

Diethylstilbestrol esters

Marketed

Major esters of diethylstilbestrol include:
Less commonly used esters of diethylstilbestrol include:
As well as the following nitrogen mustard ester:

Marketed

The following nitrogen mustard ester of hexestrol was never marketed:

Marketed

Diethylstilbestrol

Marketed