List of opioids
This is a list of opioids, opioid antagonists and inverse agonists.
[Opium] and [poppy straw] derivatives
Crude opiate extracts whole opium products
- Polish heroin
- Diascordium
- B&O Supprettes
- Dover's powder
- Kendal Black Drop
- Laudanum
- Mithridate
- Opium
- Paregoric
- Poppy straw concentrate
- Poppy tea
- Smoking opium
- Theriac
Natural opiates
Opium alkaloids
- Codeine
- Morphine
- Oripavine
- Pseudomorphine
- Thebaine
Alkaloid salts mixtures
- Pantopon
- Papaveretum
- Tetrapon
Semisynthetics including [Bentley compounds]
Morphine family
- 14-Hydroxymorphine
- 2,4-Dinitrophenylmorphine
- 6-Methyldihydromorphine
- 6-Methylenedihydrodesoxymorphine
- 6-Acetyldihydromorphine
- Azidomorphine
- Chlornaltrexamine
- Chloroxymorphamine
- Desomorphine
- Dihydromorphine
- Ethyldihydromorphine
- Hydromorphinol
- Methyldesorphine
- Morphine methylbromide
- N-Phenethylnordesomorphine
- N-Phenethyl-14-ethoxymetopon
- N-Phenethylnormorphine
- 6-Nicotinoyldihydromorphine
- RAM-378
- Ro-1539
3,6-diesters of morphine
- Acetylpropionylmorphine
- 3,6-Dibutanoylmorphine
- Diacetyldihydromorphine
- Dibutyrylmorphine
- Dibenzoylmorphine
- Diformylmorphine
- Dipropanoylmorphine
- Heroin
- Nicomorphine
Codeine-dionine family
- 6-Monoacetylcodeine
- Benzylmorphine
- Codeine methylbromide
- Desocodeine
- Dimethylmorphine
- Ethyldihydromorphine
- Methyldihydromorphine
- Ethylmorphine
- Heterocodeine
- Isocodeine
- Pholcodine
- Myrophine
- Thebacon
- Transisocodeine
Morphinones and morphols
- 14-Cinnamoyloxycodeinone
- 14-Ethoxymetopon
- 14-Methoxymetopon
- 14-Phenylpropoxymetopon
- 3-Acetyloxymorphone
- 3,14-Diacetyloxymorphone
- 7-Spiroindanyloxymorphone
- 8,14-Dihydroxydihydromorphinone
- Acetylcodone
- Acetylmorphone
- α-hydrocodol
- Benzhydrocodone
- Bromoisopropropyldihydromorphinone cas?
- Codeinone
- Codoxime
- Conorfone
- IBNtxA
- Thebacon
- Hydrocodone
- Hydromorphone
- Hydroxycodeine
- Metopon
- Morphenol
- Morphinone
- Morphol
- N-Phenethyl-14-ethoxymetopon
- Noroxymorphone
- Oxycodone
- Oxymorphol
- Oxymorphone
- Pentamorphone
- Semorphone
Morphides
- α-Chlorocodide
- β-Chlorocodide
- α-Chloromorphide
- Bromocodide
- Bromomorphide
- Chlorodihydrocodide
- Chloromorphide
- Codide
Dihydrocodeine series
- 14-Hydroxydihydrocodeine
- Acetyldihydrocodeine
- Dihydrocodeine
- Dihydrodesoxycodeine
- Dihydroisocodeine
- Nicocodeine
- Nicodicodeine
Nitrogen morphine derivatives
- 1-Nitrocodeine cas?
- Codeine-N-oxide
- Morphine-N-oxide
Hydrazones
- Oxymorphazone
Halogenated morphine derivatives
- 1-Bromocodeine
- 1-Chlorocodeine
- 1-Iodomorphine
Active opiate metabolites
- Codeine-6-glucuronide
- Codeine-N-oxide
- Heroin-7,8-oxide
- Morphine-6-glucuronide
- 3-Monoacetylmorphine
- 6-Monoacetylmorphine
- Morphine-N-oxide
- Naltrexol
- Norcodeine
- Normorphine
[Morphinan]s
Morphinan series
- 3-Hydroxymorphinan
- 4-Chlorophenylpyridomorphinan
- Cyclorphan
- Levargorphan
- Levorphanol
- Levophenacylmorphan
- Levomethorphan
- Methorphan
- Morphanol
- Norlevorphanol
- N-Methylmorphinan
- Oxilorphan
- Phenomorphan
- Proxorphan
- Ro4-1539
- Stephodeline Xorphanol
Others
- 1-Nitroaknadinine * 14-episinomenine
- 5,6-Dihydronorsalutaridine
- 6-Keto Nalbuphine
- Aknadinine
- Butorphanol
- Cephakicine
- Cephasamine
- Cyprodime
- Drotebanol
- Fenfangjine G
- Ketorfanol
- Nalbuphine
- Nalbuphone
- Tannagine
[Benzomorphan]s
- 5,9 alpha-diethyl-2-hydroxybenzomorphan
- 8-Carboxamidocyclazocine
- Alazocine
- Anazocine
- Bremazocine
- Butinazocine
- Carbazocine
- Cogazocine
- Cyclazocine
- Dezocine
- Eptazocine
- Etazocine
- Ethylketazocine
- Fedotozine
- Fluorophen
- Gemazocine
- Ibazocine
- Ketazocine
- Metazocine
- Moxazocine
- Pentazocine
- Phenazocine
- Quadazocine
- SKF-10047
- Thiazocine
- Tonazocine
- Volazocine
- Zenazocine
[4-Phenylpiperidine]s
[Pethidine]s (meperidines)
- 4-Fluoropethidine
- Allylnorpethidine
- Anileridine
- Benzethidine
- Carperidine
- Difenoxin
- Diphenoxylate
- Etoxeridine
- Furethidine
- Hydroxypethidine
- Morpheridine
- Meperidine-N-oxide
- Oxpheneridine
- Pethidine
- Pethidine intermediate A
- Pethidine intermediate B
- Pethidine intermediate C
- Pheneridine
- Phenoperidine
- Piminodine
- Properidine
- Sameridine
[Prodine]s
- Allylprodine
- -Meprodine
- Desmethylprodine
- PEPAP
- -Prodine
- Prosidol
- Trimeperidine
[Ketobemidone]s
- Acetoxyketobemidone
- Droxypropine
- Ketobemidone
- Methylketobemidone
- Propylketobemidone
Others
- Alvimopan
- Loperamide
- Picenadol
Open chain">Open-chain compound">Open chain opioids
Amidones
- Dextromethadone
- Dipipanone
- Isomethadone
- Levoisomethadone
- Levomethadone
- Methadone
- Methadone intermediate
- Normethadone
- Norpipanone
- Phenadoxone
Methadols
- Acetylmethadol
- Alphaacetylmethadol
- Alphamethadol
- Betacetylmethadol
- Betamethadol
- Dimepheptanol
- Isomethadol
- Levacetylmethadol
- Noracymethadol
Moramides
- Desmethylmoramide
- Dextromoramide
- Levomoramide
- Moramide intermediate
- Racemoramide
[Thiambutene]s
- Diethylthiambutene
- Dimethylthiambutene
- Ethylmethylthiambutene
- Piperidylthiambutene
- Pyrrolidinylthiambutene
- Thiambutene
Phenalkoxams
- Dextropropoxyphene
- Dimenoxadol
- Dioxaphetyl butyrate
- Levopropoxyphene
- Norpropoxyphene
- Pyrroliphene
Ampromides
- Diampromide
- Phenampromide
- Propiram
Others
- Embutramide
- IC-26
- Isoaminile
- Lefetamine
- R-4066
Anilidopiperidines
- 3-Allylfentanyl
- 3-Methylfentanyl
- 3-Methylthiofentanyl
- 4-Phenylfentanyl
- Alfentanil
- α-Methylacetylfentanyl
- α-Methylfentanyl
- α-Methylthiofentanyl
- Benzylfentanyl
- β-hydroxyfentanyl
- β-hydroxythiofentanyl
- β-Methylfentanyl
- Brifentanil
- Butyrfentanyl
- Carfentanil
- Fentanyl
- Lofentanil
- N-Methylcarfentanil
- Mirfentanil
- Ocfentanil
- Ohmefentanyl
- Parafluorofentanyl
- Phenaridine
- R-30490
- Remifentanil
- Sufentanil
- Thenylfentanyl
- Thiofentanyl
- Trefentanil
[Oripavine] derivatives
- 7-PET
- Acetorphine
- Alletorphine
- BU-48
- Buprenorphine
- Buprenorphine-3-glucuronide
- Cyprenorphine
- Dihydroetorphine
- Etorphine
- Homprenorphine
- 18,19-Dehydrobuprenorphine
- N-cyclopropylmethylnoretorphine
- Nepenthone
- Norbuprenorphine
- Norbuprenorphine-3-glucuronide
- Thevinone
- Thienorphine
[Phenazepane]s
- Ethoheptazine
- Meptazinol
- Metheptazine
- Metethoheptazine
- Proheptazine
Pirinitramides
- Bezitramide
- Piritramide
[Benzimidazole]s
- Clonitazene
- Etonitazene
- Isotonitazene
- Metonitazene
[Indole]s
- 18-Methoxycoronaridine
- 7-Acetoxymitragynine
- 7-Hydroxymitragynine
- ψ-Akuammigine
- Akuammidine
- Akuammine
- Coronaridine
- Eseroline
- Hodgkinsine
- Ibogaine
- Mitragynine
- Mitragynine pseudoindoxyl
- Noribogaine
- Pericine
- Pseudoakuammigine
Beta">Beta-peptide">Beta-Amino">Amine">Amino [Ketone]s
- 3--2,2-dimethyl-1-phenylpropan-1-one
[Diphenylmethylpiperazine]s
- BW373U86
- DPI-221
- DPI-287
- DPI-3290
- SNC-80
- AZD-2327
[Opioid peptide]s
[Dynorphin]s
- Big dynorphin
- Dynorphin A
- Dynorphin B
- Leumorphin
[Endomorphin]s
- Endomorphin-1
- Endomorphin-2
[Endorphin]s
- α-Endorphin
- β-Endorphin
- γ-Endorphin
- α-Neoendorphin
- β-Neoendorphin
[Enkephalin]s
- DADLE
- DAMGO
- Dermenkephalin
- Met-enkephalin
- Leu-enkephalin
Propeptides
- Proenkephalin
- Proendorphin
- Proopiomelanocortin
Others / unknown
- Adrenorphin
- Amidorphin
- Biphalin
- Casokefamide
- Casomorphins
- Cytochrophin-4
- DALDA
- Deltorphin A
- Deltorphin I
- Deltorphin II
- Deprolorphin
- Dermorphin
- DPDPE
- Frakefamide
- Gliadorphin
- Gluten exorphinss
- Hemorphin-4
- Metkefamide
- Morphiceptin
- Nociceptin
- Octreotide
- Opiorphin
- Rubiscolin
- Soymorphins
- Spinorphin
- TRIMU 5
- Tynorphin
- Valorphin
- Zyklophin
Others
- 3--3-ethoxycarbonyltropane
- AD-1211
- AH-7921
- Axomadol
- Azaprocin
- BDPC
- Bisnortilidine
- BRL-52537
- Bromadol
- Bromadoline
- Ciprefadol
- Ciramadol
- Doxpicomine
- Enadoline
- Faxeladol
- GR-89696
- Herkinorin
- ICI-199,441
- ICI-204,448
- Ketamine
- KNT-42
- LPK-26
- Lufuradom
- Metofoline
- MT-45
- Desmethylclozapine
- Nexeridine
- NNC 63-0532
- Nortilidine
- O-Desmethyltramadol
- Phenadone
- Phencyclidine
- Prodilidine
- Profadol
- Ro64-6198
- Salvinorin A
- Salvinorin B ethoxymethyl ether
- Salvinorin B methoxymethyl ether
- SB-612,111
- SC-17599
- RWJ-394,674
- TAN-67
- Tapentadol
- Thiobromadol
- Tifluadom
- Tilidine
- Tramadol
- Trimebutine
- U-47,700
- U-50,488
- U-69,593
- Viminol
- 1-piperidylidene-2-sulfonamide
Opioid antagonists">Receptor antagonist">antagonists and [inverse agonist]s
- 4-Caffeoyl-1,5-quinide
- 5'-Guanidinonaltrindole
- β-Funaltrexamine
- 6β-Naltrexol
- 6β-Naltrexol-d4
- Alvimopan
- AT-076
- Binaltorphimine
- BU09059
- Buprenorphine
- Chlornaltrexamine
- Clocinnamox
- Cyclazocine
- Cyprodime
- Diacetylnalorphine
- Diprenorphine
- Fedotozine
- ICI-174864
- J-113,397
- JDTic
- JTC-801
- Levallorphan
- LY-2456302
- LY-255582
- Methocinnamox
- Methylnaltrexone
- ML350
- Naldemedine
- Nalfurafine
- Nalmefene
- Nalmexone
- Nalodeine
- Naloxazone
- Naloxegol
- Naloxol
- Naloxonazine
- Naloxone
- Naloxone benzoylhydrazone
- Nalorphine
- Naltrexone
- Naltriben
- Naltrindole
- Norbinaltorphimine
- Oxilorphan
- PF-4455242
- S-allyl-3-hydroxy-17-thioniamorphinan
- Samidorphan
- SR-16430
Biased ligands">Functional selectivity">Biased ligands
- 6'-Guanidinonaltrindole
- 7-Hydroxymitragynine
- Herkinorin
- ICI-199,441
- Noribogaine
- Oliceridine
- RB-64
- TRV734
Receptor heteromer">GPCR oligomer">Receptor heteromer targeting ligands
- 6'-GNTI
- CYM-51010
- NNTA
- IBNtxA
Uncategorized opioids
- ADL-5859
- Alimadol
- Amentoflavone
- Anilopam
- Asimadoline
- Cyproterone acetate
- FE 200665
- Fedotozine
- HZ-2
- Kolokol-1
- Matrine
- MCOPPB
- Menthol
- MT-7716
- Nalfurafine
- Nalorphine
- Nalorphine dinicotinate
- PZM21
- Proglumide
- Ro65-6570
- SoRI-9409
- Spiradoline
- SR-8993
- SR-16435
Combination drug formulations containing opioids
- Buprenorphine/naloxone
- Buprenorphine/samidorphan
- Bupropion/naltrexone
- Co-codamol
- Co-codaprin
- Co-dydramol
- Co-proxamol
- Fentanyl/fluanisone
- Hydrocodone/ibuprofen
- Hydrocodone/paracetamol
- Loperamide/simethicone
- Morphine/naltrexone
- Oxycodone/aspirin
- Oxycodone/naloxone
- Oxycodone/paracetamol